From: PI3Kγδ inhibition suppresses key disease features in a rat model of asthma
Compound
Human ppb (fu, %)
Human plasma fu
Fu’
PI3Kγδ - AZD8154
0.63
0.0063
0.060
PI3Kδ - GSK2269557
2.1
0.021
0.177
PI3Kγ - AZD3458
15
0.15
0.638