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Table 1 Relative receptor affinities of mometasone furoate (MF, data from [7]), its metabolites 6β-hydroxy mometasone furoate (6β-OH MF), mometasone and the major degradation product 9,11-epoxy mometasone furoate (9,11-epoxy MF) in relation to dexamethasone (Dexa). Values represent mean and mean deviation of the mean of n = 3 independent experiments.

From: Significant receptor affinities of metabolites and a degradation product of mometasone furoate

Compound

Relative receptor affinity (RRA)

Mean deviation of the mean

MF

2244

± 142

Dexa

100

± 10

6β-OH MF

206

± 15

9,11-epoxy MF

220

± 22

Mometasone

781

± 27